Liphello tsa Meriana ea Bohloko le Thibelo ea Matšoao a ho Furalla
Buprenorphine e ka sehlopheng sa meriana e bitsoang li-opioid tse hanyetsanang le li-agonist. E sebelisoa litšoantšong tse fetisisang le lifilimi tsa batho ba hlokang meriana ea ho pota-pola mahlaba bakeng sa bohloko bo ke keng ba phekoloa ka meriana e meng. E boetse e sebelisoa ho thibela matšoao a ho tlohela bakuli ba khaotsang ho sebelisa lithethefatsi tsa opioid ka ho hlahisa lithethefatsi tsena tse tšoanang.
Buprenorphine e boetse e tsejoa e le Suboxone (buprenorphine le naloxone), Subutex, Belbuca, Buprenex, Butrans, Temgesic, le Bupe
Ho ithuta hore na e sebetsa joang tsamaisong ea hau le hore na ho kopana ho ka bang le lithethefatsi tse ling ho ka thusa ho utloisisa mekhoa ea ho qoba le ho thibela ho feta tekano.
Buprenorphine ho Tsamaiso ea hau
Buprenorphine ke opioid e matla, e tšoarellang nako e telele esita le haeba u e nka ho ea ka litaelo tsa ngaka ea hao, u tlameha ho hlahlojoa ka ho khoneha hore u itšoare ka matla, haholo-holo ha u nka buprenorphine pele kapa ha tekanyo e fetoha.
Websaete ea FDA e na le Litlhahiso tsa Meriana bakeng sa mabitso a mangata a lihlahisoa tsa buprenorphine. U lokela ho botsa ngaka ea hau kapa lihlopha tsena bakeng sa mehato e tobileng ea ho itšireletsa, lithibelo le tlhahiso-leseling e eketsehileng bakeng sa sehlahisoa se seng le se seng.
Litla-morao tsa buprenorphine li fumaneha ka har'a li-receptor tse bohloko tsa bokopi bokong le mokokong oa mokokotlo. Empa hape e nyahamisa litsi tsa phefumoloho tsa boko.
E hlahisa bana ba pinpoint. E fokotsa motility ea mongobo, e leng se ka lebisang ho tiisetsoa. Hape ke vasodilator mme kahoo e ka hlahisa letlalo le tsitsitseng, ho fufuleloa le ho nyahama ha u tsoha ka mor'a ho robala kapa ho lula.
Buprenorphine e na le nako e telele ea bophelo ba lihora tse 24 ho isa ho tse 42. E robehile ke sebete 'me e fetiselitsoe ka bile le liphio ka hara moroto le li-feces.
Bakeng sa motsoako oa Suboxone, naloxone e na le nako e khutšoanyane ea ho felisa ka nako ea ho felisa bophelo ba lihora tse peli ho isa ho tse 12.
Ho na le litšebelisano tse ngata tsa lithethefatsi le buprenorphine tse ka lebisang liketsong tse matla le mohlomong tse bolaeang. U se ke ua noa joala kapa ua noa meriana leha e le efe e akarelletsang ho noa joala ho noa buprenorphine. U se ke ua nka lithethefatsi tsa seterateng.
Ha u ntse u hloka ho bua ka meriana eohle, li-supplement, li-vithamine le lithethefatsi tse ngata ho feta ngaka ea hau, tsena ke tsona tse amehang ka ho fetisisa: benzodiazepines (e kang Xanax, Librium, Klonopin, Valium, Diastat, Ativan, Restoril, Halcion le bohle ba bang), li-relaxation tsa mesifa, li-sedative, lipilisi tse robalang, li-tranquilizers, meriana e bohloko, le meriana ea mafu a kelello le ho nyeheloa ke pelo.
Haeba u khaotsa ho sebelisa buprenorphine ka tšohanyetso, u ka 'na ua ba le matšoao a ho khaotsa.
Ho thibela ho feta ha Buprenorphine
Matšoao a ho feta ho feta buprenorphine a ka kenyeletsa:
- Sheba bana
- Ho otsela haholo
- Sehlōhō
- Pono e fosahetseng
- Ho fokola ho fokola
Haeba u belaella hore motho e mong o fetetse ho feta buprenorphine, letsetsa setsing sa thibelo ea chefo ho 1-800-222-1222. Haeba motho ea hlokofalitsoeng a oa kapa a sa heme, founa 9-1-1.
Buprenorphine e telele e lutse joang tsamaisong ena
Ho leka ho lekanya hantle hore na buprenorphine e ka fumanoa nako e telele hakae 'meleng ho itšetlehile ka mefuta e mengata, ho kenyelletsa le mofuta ofe oa tlhahiso ea lithethefatsi e sebelisitsoeng, ebang e kopane le lithethefatsi tse ling, le metabolism ka bomong.
Buprenorphine e na le metabolite (norbuprenorphine) e fapaneng ho feta e tloaelehileng ea opioids mme e ka 'na ea se ke ea lekoa bakeng sa lisebelisoa tsa lithethefatsi tsa moroto tse sebelisetsoang mosebetsi. Leha ho le joalo, tlhahlobo ea eona e se e tloaelehile haholoanyane. Haeba o laetsoe buprenorphine kapa sehlahisoa sa Suboxone, o lokela ho se senolela le laborateng ea teko e le hore litholoana tsa hau li ka hlalosoa hantle. E ka fumanoa ka metsing ka matsatsi a 6, empa le ho feta ho latela metabolism. E ka fumanoa ho skrine ea urine ea opioid e loantšitsoeng kapa skrine e itseng ea buprenorphine ea urine.
> Mehloli:
> Boitsebiso ba lithethefatsi ba Buprenorphine. Redwood Toxicology Laboratory. https://www.redwoodtoxicology.com/resources/drug_info/buprenorphine.
> Buprenorphine Buccal (bohloko bo sa foleng). Medline Plus NIH. https://medlineplus.gov/druginfo/meds/a616019.html.
> Buprenorphine Sublingual le Buccal (ho itšetleha ka opioid). Medline Plus NIH. https://medlineplus.gov/druginfo/meds/a605002.html.
> Buprenorphine Transdermal Patch. Medline Plus NIH. https://medlineplus.gov/druginfo/meds/a613042.html.