Modafinil (Provigil) e sebelisetsoa ho tšoaroa ke ho robala ha boroko, ho hlajoa ke pelo le ho feta.
Batho ba bangata ba sebelisa hampe lithethefatsi tse matlafatsang kapa tsa psychosotimulant boemong bo sa ngolisoeng ho ngola hore ho eketsa tlhahiso, ho loantša mokhathala le thuso ka mathata a kelello. Le hoja ho sebelisoa hampe ka lithethefatsi tse matlafatsang tse kang amphetamine, methylphenidate, le modafinil (Provigil) ka tloaelo li amahanngoa le liithuti tsa univesithing - ho hakanyetsoa hore karolo ea 7 ho isa ho 20 lekholong ea liithuti tsa univesithi tsa United States li tlalehile hore li sebelisa lithethefatsi hampe - lihlopha tse ling tse makatsang tsa batho ba li sebelisa hampe lithethefatsi, hape.
Ka mohlala, karolo ea 8,9 lekholong ea lingaka tse buoang tse entsoeng Jeremane e tlalehile hore ho se sebelisoe ka mokhoa o ngotsoeng oa lithethefatsi tse matlafatsang.
Modafinil e tlameha ho se be lemallo ho feta tse ling tsa psychostimulants tse kang amphetamine; Leha ho le joalo, re ntse re sa utloisise hantle hore na lithethefatsi tsena li sebetsa joang kapa liphello tsa nako e telele hakae. Ho feta moo, modafinil e ka baka liphello tse ling tse tebileng tse mpe 'me e lokela ho nkoa feela ha e ngotsoe ke ngaka.
Modafinil ke eng?
Ka linako tse ling Modafinil e bitsoa "moemeli oa ho tsosa ka matla." Bafuputsi ba lumela hore lithethefatsi tsena li sebetsa ka ho eketsa ho fumaneha ha synaptic ea li-neurotransmitters tse kang monoamines, catecholamines, dopamine, serotonin, adenosine, histamine le noradrenaline. Modafinil e ama hypothalamus, hippocampus, le amygdala tseo e leng likarolo tsa boko.
Modafinil ke letlapa le nkiloeng ka molomo hangata ka letsatsi. Batho ba bangata ba sebetsang motšehare ba noa lithethefatsi hoseng ho sa tsotellehe malapa a feletseng kapa a se nang letho. Leha ho le joalo, basebetsi ba nkang lithethefatsi ho tsosolosa ho tsoha ba noa meriana pele lifofane li qala.
Modafinil e Tšoara Eng?
Modafinil e sebelisetsoa ho sebetsana le mathata ka kutloisiso, ho tsosoa le ho tsoha. Maemo a mang a tšoaroang ka modafinil a akaretsa tse latelang:
- Ho senyeha ha maikutlo
- Sebetsa-ho sebetsana le bothata ba ho robala
- Ho thibela ho robala ha boroko
- Kotsi e mpe ea boko
- Phekolo ea lefu la ho tepella maikutlo
- ADHD
- Tlhokomelo ea ho qetela kapa ea ho qetela ea bophelo
Mabapi le tlhokomelo e fokolang kapa ea ho qetela ea bophelo, litsebi tse ngata li khetha ho beha li-psycho-stimulants joaloka modafinil hobane li ntlafatsa mehopolo ho feta meriana ea mafu a kelello. Ho feta moo, ho itšetleha ha ho na tlhokomelo e fokolang nakong ea tlhokomelo ea ho qetela ea bophelo.
Liphello tse mpe
Liphetho tse bohloko tse tloaelehileng tsa Modafinil li kenyeletsa tse latelang:
- Ho otla
- Nausea
- Ho tsitlella
- Ho tšoenyeha
Liphetho tse ling tse bohloko li kenyeletsa tse latelang:
- Ho tsieleha
- Letšollo
- Ho tlosoa ha 'mele
- Ho rohakana
- Hoarseness
- Ho phefumoloha ho thata
- Mahlaba a sefuba
- Ho otlolla pelo ho sa tloaelehang
- Maikutlo a ho ipolaea (menahano ea ho ipolaea)
- Hallucination
- Rash
- Blisters
- Hives
Tse ling tsa liphello tsena tse bohloko li tšosoa ebile lia kotsi, e-ba bonnete ba hore u ikopanye le ngaka ea hau haeba u e-na le e 'ngoe ea tsona.
Ho phaella moo, tse ling tsa liphello tse bohloko tse kang ho hlobaela, ho hloka botsitso, bohloko ba sefuba, ho nyekeloa ke pelo, le pherekano li ka bakoa ke ho feta tekano ka modafinil. Haeba u belaella ho fetela holimo, letsetsa lits'ebeletso tsa tšohanyetso kapa u iteanye le ngaka hang-hang.
Litlhōlisano
Modafinil ha e mong le e mong, mme pele ngaka ea hau e u laela meriana ena, o lokela ho mo tsebisa tse latelang:
- Ho tsuba ho modafinil kapa armodafinil (enantiomeri ea modafinil)
- Meriana e imetsoeng kelellong e kenyelletsang SSRIs, TCAs le benzodiazepines
- Ho noa meriana e kang phenytoin le carbamazepine
- Meriana e mengata joaloka itraconazole le ketoconazole
- Tšebeliso e mpe ea lithethefatsi kapa ho itšetleha ka eona
- Li-vithamine, li-supplement le phepo e nepahetseng
Batho ba nang le angina kapa ba sa tsoa ba le lefu la pelo ha baa lokela ho fuoa modafinil. Ho feta moo, ha ho hlaka hore na modafinil e na le phello e kae moeling oa maqheku. Kahoo, modafinil e ka ba kotsi ho batho ba nang le lefu la sethoathoa le mathata a mang a ho tšoaroa ke lefu.
Ha ho na lithuto tsa nako e telele liphello tsa modafinil bokong. Ngaka e lokela ho hlahloba ka hloko hore na e ka fana ka modafinil le ho lekanya molemo oa thepa ea eona e susumetsang e nang le liphello tse mpe.
Le hoja modafinil mohlomong e sa lemalla ho feta tse ling tse susumetsang joaloka amphetamines le methylphenidate, e ntse e ka etsa hore motho a itšetlehe ka eona.
Ka kōpo utloisisa hore nako le nako ha ngaka e etsa qeto ea ho beha modafinil, qeto ena ke e fanang ka mamello. Ka mantsoe a mang, haeba u laetsoe modafinil kapa psychostimulant efe kapa efe, lengolo lena la ngaka ke lona feela. Ha ua lokela ho arolelana kapa ho rekisa modafinil-kapa lithethefatsi leha e le life tsa ngaka bakeng sa taba eo. Ho itokolla ho joalo ho kotsi ebile ha ho molaong.
Lisebelisoa
Liu D, Norman MA, Singh B, Lee K. Ho tepella maikutlo le Tse ling tsa Litaba tsa Bophelo ba Mental. Ka: Williams BA, Chang A, Ahalt C, Chen H, Conant R, Landefeld C, Ritchie C, Yukawa M. eds. Tlhahlobo ea Hona joale le Phekolo: Geriatrics, Second Edition . New York, NY: Hill ea McGraw; 2014.
Siu G. Pharmacotherapy. Ka: Maitin IB, Cruz E. eds. Tlhaloso ea CURRENT & Tlhokomelo: Meriana ea 'mele le ho tsosolosoa . New York, NY: Hill ea McGraw; 2015.
Sehlooho se nang le sehlooho se reng, "Ho sebelisoa ha basebetsi ba thuto ea litsebi tsa New Zealand" ho ba le likhallelo tse ngata tse nang le ts'ebeliso ea likhopolo-taba "S Ram le li-co-author tsa Drug le Alcohol Review e hatisitsoeng ka 2015.